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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA RECQL4 GDSC1000 pan-cancer AAC 0.091 0.005
mRNA FAM43B CTRPv2 pan-cancer AAC 0.1 0.005
mRNA PDPK1 GDSC1000 pan-cancer AAC -0.09 0.005
mRNA DIAPH1 CTRPv2 pan-cancer AAC 0.11 0.005
mRNA ARG2 GDSC1000 pan-cancer AAC 0.094 0.005
mRNA MMS19 CTRPv2 pan-cancer AAC 0.1 0.005
mRNA MED8 CTRPv2 pan-cancer AAC -0.1 0.005
mRNA ZNF33A CTRPv2 pan-cancer AAC 0.11 0.005
mRNA OSBPL3 GDSC1000 pan-cancer AAC -0.096 0.005
mRNA B4GALT6 GDSC1000 pan-cancer AAC -0.092 0.005
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