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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA GBGT1 GDSC1000 pan-cancer AAC 0.19 2e-09
mRNA SENP7 GDSC1000 pan-cancer AAC 0.2 3e-09
mRNA TRAK2 CTRPv2 pan-cancer AAC 0.23 4e-09
mRNA GYPA GDSC1000 pan-cancer AAC 0.18 4e-09
mRNA MYO18B GDSC1000 pan-cancer AAC 0.19 4e-09
mRNA CRADD GDSC1000 pan-cancer AAC 0.19 4e-09
mRNA SLC4A1 CTRPv2 pan-cancer AAC 0.2 4e-09
mRNA YPEL4 CTRPv2 pan-cancer AAC 0.21 4e-09
mRNA PLPPR3 GDSC1000 pan-cancer AAC 0.19 5e-09
mRNA ADAMTS14 CTRPv2 pan-cancer AAC 0.21 6e-09
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