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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA KLF1 CTRPv2 pan-cancer AAC 0.22 9e-10
mRNA KEL GDSC1000 pan-cancer AAC 0.2 1e-09
mRNA KIAA1586 GDSC1000 pan-cancer AAC 0.21 1e-09
mRNA SLC6A19 CTRPv2 pan-cancer AAC 0.22 1e-09
mRNA CEP57L1 GDSC1000 pan-cancer AAC 0.2 1e-09
mRNA N4BP2 CTRPv2 pan-cancer AAC 0.24 1e-09
mRNA RHD GDSC1000 pan-cancer AAC 0.19 1e-09
mRNA PIM1 GDSC1000 pan-cancer AAC 0.2 1e-09
mRNA ZNF627 GDSC1000 pan-cancer AAC 0.2 2e-09
mRNA AC104389.2 CTRPv2 pan-cancer AAC 0.21 2e-09
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