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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA GOLGA8J CTRPv2 pan-cancer AAC 0.23 3e-10
mRNA MLC1 GDSC1000 pan-cancer AAC 0.22 3e-10
mRNA ABL1 GDSC1000 pan-cancer AAC 0.21 3e-10
mRNA NFE2 CTRPv2 pan-cancer AAC 0.24 4e-10
mRNA EGFL7 GDSC1000 pan-cancer AAC 0.2 4e-10
mRNA IKZF4 CTRPv2 pan-cancer AAC 0.24 5e-10
mRNA TAS2R5 CTRPv2 pan-cancer AAC 0.23 5e-10
mRNA HEMGN GDSC1000 pan-cancer AAC 0.2 7e-10
mRNA SLC2A4 CTRPv2 pan-cancer AAC 0.22 8e-10
mRNA RFESD CTRPv2 pan-cancer AAC 0.23 8e-10
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