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canertinib

Synonyms

SourcesNames Used
CTRPv2canertinib
PharmacoGx canertinib

External IDs

DatabaseIdentifier
Smiles: Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Pubchem: 156414

Annotated Targets

ERBB4, EGFR, ERBB2, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to canertinib


Feature TypeStandardized
Nominal ANOVA
mRNA MKNK1 CTRPv2 pan-cancer AAC 0.15 7e-05
mRNA C1orf64 CTRPv2 pan-cancer AAC 0.15 7e-05
mRNA ARL2-SNX15 CTRPv2 pan-cancer AAC -0.14 8e-05
mRNA TCAP CTRPv2 pan-cancer AAC 0.14 8e-05
mRNA UHRF1BP1L CTRPv2 pan-cancer AAC -0.15 8e-05
mRNA TMEM254 CTRPv2 pan-cancer AAC 0.16 8e-05
mRNA FANK1 CTRPv2 pan-cancer AAC 0.15 8e-05
mRNA AC136612.1 CTRPv2 pan-cancer AAC -0.15 9e-05
mRNA TSPAN6 CTRPv2 pan-cancer AAC 0.16 9e-05
mRNA HLTF CTRPv2 pan-cancer AAC -0.14 9e-05
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