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canertinib

Synonyms

SourcesNames Used
CTRPv2canertinib
PharmacoGx canertinib

External IDs

DatabaseIdentifier
Smiles: Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Pubchem: 156414

Annotated Targets

ERBB4, EGFR, ERBB2, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to canertinib


Feature TypeStandardized
Nominal ANOVA
mRNA TMPRSS11E CTRPv2 pan-cancer AAC 0.17 2e-06
mRNA ARRDC1 CTRPv2 pan-cancer AAC 0.2 2e-06
mRNA TRPM4 CTRPv2 pan-cancer AAC 0.19 2e-06
mRNA CTSV CTRPv2 pan-cancer AAC 0.19 2e-06
mRNA CCDC77 CTRPv2 pan-cancer AAC -0.18 2e-06
mRNA RP4-777O23.3 CTRPv2 pan-cancer AAC 0.19 2e-06
mRNA TTC33 CTRPv2 pan-cancer AAC -0.17 2e-06
mRNA TSPAN1 CTRPv2 pan-cancer AAC 0.18 3e-06
mRNA COMT CTRPv2 pan-cancer AAC 0.17 3e-06
mRNA ELMO3 CTRPv2 pan-cancer AAC 0.21 3e-06
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