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canertinib

Synonyms

SourcesNames Used
CTRPv2canertinib
PharmacoGx canertinib

External IDs

DatabaseIdentifier
Smiles: Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Pubchem: 156414

Annotated Targets

ERBB4, EGFR, ERBB2, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to canertinib


Feature TypeStandardized
Nominal ANOVA
mRNA SART1 CTRPv2 pan-cancer AAC -0.084 0.02
mRNA C2CD4A CTRPv2 pan-cancer AAC -0.082 0.02
mRNA VAMP4 CTRPv2 pan-cancer AAC -0.086 0.02
mRNA PIGG CTRPv2 pan-cancer AAC 0.085 0.02
mRNA RTP2 CTRPv2 pan-cancer AAC 0.081 0.02
mRNA MANEAL CTRPv2 pan-cancer AAC -0.086 0.02
mRNA POLR2F CTRPv2 pan-cancer AAC -0.092 0.02
mRNA MAP3K12 CTRPv2 pan-cancer AAC -0.092 0.02
mRNA SLCO2B1 CTRPv2 pan-cancer AAC -0.084 0.02
mRNA NDUFB7 CTRPv2 pan-cancer AAC -0.082 0.02
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