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canertinib

Synonyms

SourcesNames Used
CTRPv2canertinib
PharmacoGx canertinib

External IDs

DatabaseIdentifier
Smiles: Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Pubchem: 156414

Annotated Targets

ERBB4, EGFR, ERBB2, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to canertinib


Feature TypeStandardized
Nominal ANOVA
mRNA SDCBP CTRPv2 pan-cancer AAC -0.093 0.02
mRNA C8G CTRPv2 pan-cancer AAC -0.083 0.02
mRNA CEBPA CTRPv2 pan-cancer AAC 0.084 0.02
mRNA REXO2 CTRPv2 pan-cancer AAC -0.085 0.02
mRNA CTU2 CTRPv2 pan-cancer AAC -0.083 0.02
mRNA FGD1 CTRPv2 pan-cancer AAC -0.094 0.02
mRNA UNC13B CTRPv2 pan-cancer AAC -0.085 0.02
mRNA NUMBL CTRPv2 pan-cancer AAC -0.089 0.02
mRNA NAA11 CTRPv2 pan-cancer AAC -0.085 0.02
mRNA ZNF547 CTRPv2 pan-cancer AAC 0.085 0.02
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