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canertinib

Synonyms

SourcesNames Used
CTRPv2canertinib
PharmacoGx canertinib

External IDs

DatabaseIdentifier
Smiles: Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Pubchem: 156414

Annotated Targets

ERBB4, EGFR, ERBB2, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to canertinib


Feature TypeStandardized
Nominal ANOVA
mRNA DHX57 CTRPv2 pan-cancer AAC -0.089 0.02
mRNA POLR1E CTRPv2 pan-cancer AAC -0.089 0.02
mRNA TMEM65 CTRPv2 pan-cancer AAC 0.086 0.02
mRNA PATE2 CTRPv2 pan-cancer AAC -0.09 0.02
mRNA CACNA2D1 CTRPv2 pan-cancer AAC -0.092 0.02
mRNA ARL5A CTRPv2 pan-cancer AAC -0.091 0.02
mRNA ZNF625 CTRPv2 pan-cancer AAC -0.096 0.02
mRNA CIAO1 CTRPv2 pan-cancer AAC -0.087 0.02
mRNA UBIAD1 CTRPv2 pan-cancer AAC -0.092 0.02
mRNA KLF8 CTRPv2 pan-cancer AAC 0.088 0.02
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