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canertinib

Synonyms

SourcesNames Used
CTRPv2canertinib
PharmacoGx canertinib

External IDs

DatabaseIdentifier
Smiles: Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Pubchem: 156414

Annotated Targets

ERBB4, EGFR, ERBB2, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to canertinib


Feature TypeStandardized
Nominal ANOVA
mRNA DUSP19 CTRPv2 pan-cancer AAC -0.15 5e-05
mRNA LMBR1 CTRPv2 pan-cancer AAC -0.15 5e-05
mRNA MPZL2 CTRPv2 pan-cancer AAC 0.16 5e-05
mRNA TRPV2 CTRPv2 pan-cancer AAC -0.17 5e-05
mRNA ARAP2 CTRPv2 pan-cancer AAC 0.15 5e-05
mRNA TMEM79 CTRPv2 pan-cancer AAC 0.16 5e-05
mRNA LYPD3 CTRPv2 pan-cancer AAC 0.16 5e-05
mRNA SLC39A14 CTRPv2 pan-cancer AAC -0.15 5e-05
mRNA KRT7 CTRPv2 pan-cancer AAC 0.16 6e-05
mRNA SPRYD7 CTRPv2 pan-cancer AAC -0.15 6e-05
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