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canertinib

Synonyms

SourcesNames Used
CTRPv2canertinib
PharmacoGx canertinib

External IDs

DatabaseIdentifier
Smiles: Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Pubchem: 156414

Annotated Targets

ERBB4, EGFR, ERBB2, AKT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to canertinib


Feature TypeStandardized
Nominal ANOVA
mRNA PAK6 CTRPv2 pan-cancer AAC 0.17 2e-05
mRNA EXOSC10 CTRPv2 pan-cancer AAC -0.16 2e-05
mRNA RAB25 CTRPv2 pan-cancer AAC 0.19 2e-05
mRNA HMGN4 CTRPv2 pan-cancer AAC -0.16 2e-05
mRNA STXBP1 CTRPv2 pan-cancer AAC -0.17 2e-05
mRNA GRB7 CTRPv2 pan-cancer AAC 0.16 2e-05
mRNA COPS8 CTRPv2 pan-cancer AAC -0.16 2e-05
mRNA MAP3K9 CTRPv2 pan-cancer AAC 0.18 2e-05
mRNA GSDMB CTRPv2 pan-cancer AAC 0.15 2e-05
mRNA SLC15A2 CTRPv2 pan-cancer AAC 0.16 2e-05
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