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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA TMEM167B GDSC1000 pan-cancer AAC -0.078 0.007
mRNA KCNH3 CTRPv2 pan-cancer AAC 0.088 0.007
mRNA DBX2 CTRPv2 pan-cancer AAC 0.091 0.007
mRNA ILK GDSC1000 pan-cancer AAC -0.081 0.007
mRNA TRIM28 CTRPv2 pan-cancer AAC 0.089 0.007
mRNA KCNN3 GDSC1000 pan-cancer AAC -0.083 0.007
mRNA COQ8A CTRPv2 pan-cancer AAC 0.098 0.007
mRNA HEXB GDSC1000 pan-cancer AAC -0.087 0.007
mRNA MYADML2 CTRPv2 pan-cancer AAC 0.085 0.007
mRNA KDSR GDSC1000 pan-cancer AAC 0.082 0.007
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