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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA SH3BP1 CTRPv2 pan-cancer AAC 0.19 2e-07
mRNA ARFGEF2 CTRPv2 pan-cancer AAC -0.16 9e-07
mRNA STAU1 CTRPv2 pan-cancer AAC -0.16 7e-06
mRNA PTP4A3 CTRPv2 pan-cancer AAC 0.15 8e-06
mRNA PDZD11 CTRPv2 pan-cancer AAC -0.16 8e-06
mRNA SPN CTRPv2 pan-cancer AAC 0.2 8e-06
mRNA ATOX1 CTRPv2 pan-cancer AAC -0.17 9e-06
mRNA AURKA CTRPv2 pan-cancer AAC -0.15 9e-06
mRNA HNRNPA1 CTRPv2 pan-cancer AAC 0.16 2e-05
mRNA MANBAL CTRPv2 pan-cancer AAC -0.18 2e-05
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