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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA TFAP4 CTRPv2 pan-cancer AAC 0.14 0.0002
mRNA MTR GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA CREB1 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA EMID1 CTRPv2 pan-cancer AAC 0.12 0.0002
mRNA JMJD1C GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA PTBP2 GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA SQSTM1 GDSC1000 pan-cancer AAC -0.12 0.0002
mRNA KHSRP GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA CYP4F22 GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA MYC GDSC1000 pan-cancer AAC 0.12 0.0002
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