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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA ITGA2B GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA PTPN7 GDSC1000 pan-cancer AAC 0.18 0.0002
mRNA TYK2 CTRPv2 pan-cancer AAC 0.16 0.0002
mRNA NACA2 GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA KDM2B GDSC1000 pan-cancer AAC 0.13 0.0002
mRNA PAXBP1 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA LMO2 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA CD163 GDSC1000 pan-cancer AAC -0.1 0.0002
mRNA TRIM33 GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA ZRANB2 GDSC1000 pan-cancer AAC 0.12 0.0002
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