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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA FAM167A GDSC1000 pan-cancer AAC -0.11 0.0001
mRNA BRI3 GDSC1000 pan-cancer AAC -0.11 0.0002
mRNA TJP1 GDSC1000 pan-cancer AAC -0.21 0.0002
mRNA SIAH3 GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA S1PR4 GDSC1000 pan-cancer AAC 0.15 0.0002
mRNA FTL GDSC1000 pan-cancer AAC -0.11 0.0002
mRNA CYTL1 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA HMGB1 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA CD109 GDSC1000 pan-cancer AAC -0.12 0.0002
mRNA CTR9 GDSC1000 pan-cancer AAC 0.11 0.0002
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