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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA GYPE GDSC1000 pan-cancer AAC 0.11 9e-05
mRNA MTG2 CTRPv2 pan-cancer AAC -0.13 9e-05
mRNA DAB1 GDSC1000 pan-cancer AAC 0.12 9e-05
mRNA RNF220 GDSC1000 pan-cancer AAC 0.11 9e-05
mRNA HSD3B7 GDSC1000 pan-cancer AAC -0.12 9e-05
mRNA HNRNPM GDSC1000 pan-cancer AAC 0.12 9e-05
mRNA TRIM10 GDSC1000 pan-cancer AAC 0.11 0.0001
mRNA KDM3B GDSC1000 pan-cancer AAC 0.12 0.0001
mRNA SMARCC1 CTRPv2 pan-cancer AAC 0.14 0.0001
mRNA EDRF1 GDSC1000 pan-cancer AAC 0.12 0.0001
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