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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA BIN2 CTRPv2 pan-cancer AAC 0.1 0.007
mRNA USF3 GDSC1000 pan-cancer AAC 0.077 0.007
mRNA DRAXIN GDSC1000 pan-cancer AAC 0.076 0.007
mRNA RBPMS2 CTRPv2 pan-cancer AAC 0.088 0.007
mRNA LRRC8B GDSC1000 pan-cancer AAC 0.086 0.007
mRNA LRRC4C GDSC1000 pan-cancer AAC 0.085 0.007
mRNA CRELD1 GDSC1000 pan-cancer AAC -0.079 0.007
mRNA CMC2 GDSC1000 pan-cancer AAC -0.076 0.007
mRNA DLAT GDSC1000 pan-cancer AAC 0.079 0.007
mRNA CERCAM GDSC1000 pan-cancer AAC -0.081 0.007
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