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TPCA-1

Synonyms

SourcesNames Used
GDSC1000, CTRPv2TPCA-1
PharmacoGx TPCA-1

External IDs

DatabaseIdentifier
Smiles: NC(=O)Nc1sc(cc1C(=O)N)c2ccc(F)cc2
Pubchem: 9903786

Annotated Targets

IKBKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to TPCA-1


Feature TypeStandardized
Nominal ANOVA
mRNA EWSR1 CTRPv2 pan-cancer AAC 0.094 0.006
mRNA NABP1 CTRPv2 pan-cancer AAC -0.089 0.006
mRNA MYH15 CTRPv2 pan-cancer AAC -0.088 0.006
mRNA SESTD1 CTRPv2 pan-cancer AAC 0.092 0.006
mRNA NPC1L1 CTRPv2 pan-cancer AAC 0.092 0.006
mRNA ABCC2 GDSC1000 pan-cancer AAC -0.081 0.006
mRNA KAT6A GDSC1000 pan-cancer AAC 0.084 0.006
mRNA KRTAP6-3 CTRPv2 pan-cancer AAC -0.086 0.006
mRNA C19orf35 CTRPv2 pan-cancer AAC 0.091 0.006
mRNA TBX5 CTRPv2 pan-cancer AAC 0.093 0.006
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