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GMX-1778

Synonyms

SourcesNames Used
CTRPv2GMX-1778
PharmacoGx GMX-1778

External IDs

DatabaseIdentifier
Smiles: Clc1ccc(OCCCCCCN=C(NC#N)Nc2ccncc2)cc1

Annotated Targets

NAMPT

FDA Approval Status

Not Approved
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Top molecular features associated with response to GMX-1778


Feature TypeStandardized
Nominal ANOVA
mRNA SHISA8 CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA DLL1 CTRPv2 pan-cancer AAC 0.13 0.0004
mRNA MALL CTRPv2 pan-cancer AAC -0.14 0.0004
mRNA POLR1D CTRPv2 pan-cancer AAC 0.14 0.0004
mRNA HTT CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA CNTNAP2 CTRPv2 pan-cancer AAC 0.13 0.0004
mRNA TEX13B CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA EEF1E1-BLOC1S5 CTRPv2 pan-cancer AAC 0.13 0.0004
mRNA MAPK8IP2 CTRPv2 pan-cancer AAC 0.14 0.0004
mRNA CBR1 CTRPv2 pan-cancer AAC -0.13 0.0004
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