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TG-101348

Synonyms

SourcesNames Used
GDSC1000TG101348
CTRPv2TG-101348
PharmacoGx TG-101348

External IDs

DatabaseIdentifier
Smiles: CC1=CN=C(N=C1NC2=CC(=CC=C2)S(=O)(=O)NC(C)(C)C)NC3=CC=C(C=C3)OCCN4CCCC4
Inchikey: JOOXLOJCABQBSG-UHFFFAOYSA-N
Pubchem: 16722836

Annotated Targets

BRD4, JAK1, JAK2, JAK3, TYK2

FDA Approval Status

Not Approved
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Top molecular features associated with response to TG-101348


Feature TypeStandardized
Nominal ANOVA
mRNA MYB GDSC1000 pan-cancer AAC 0.28 5e-12
mRNA GMFG GDSC1000 pan-cancer AAC 0.28 6e-08
mRNA NCKAP1L GDSC1000 pan-cancer AAC 0.26 3e-08
mRNA PTPN7 GDSC1000 pan-cancer AAC 0.23 8e-07
mRNA SPN CTRPv2 pan-cancer AAC 0.22 8e-07
mRNA LAIR1 GDSC1000 pan-cancer AAC 0.22 3e-09
mRNA GMFG CTRPv2 pan-cancer AAC 0.21 5e-06
mRNA MFNG GDSC1000 pan-cancer AAC 0.21 1e-05
mRNA FLT3 GDSC1000 pan-cancer AAC 0.21 5e-13
mRNA MYB CTRPv2 pan-cancer AAC 0.21 8e-07
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