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TG-101348

Synonyms

SourcesNames Used
GDSC1000TG101348
CTRPv2TG-101348
PharmacoGx TG-101348

External IDs

DatabaseIdentifier
Smiles: CC1=CN=C(N=C1NC2=CC(=CC=C2)S(=O)(=O)NC(C)(C)C)NC3=CC=C(C=C3)OCCN4CCCC4
Inchikey: JOOXLOJCABQBSG-UHFFFAOYSA-N
Pubchem: 16722836

Annotated Targets

BRD4, JAK1, JAK2, JAK3, TYK2

FDA Approval Status

Not Approved
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Top molecular features associated with response to TG-101348


Feature TypeStandardized
Nominal ANOVA
mRNA CMC4 CTRPv2 pan-cancer AAC -0.14 5e-05
mRNA CTBP2 GDSC1000 pan-cancer AAC 0.15 5e-05
mRNA GNA15 GDSC1000 pan-cancer AAC 0.13 5e-05
mRNA POLR3G CTRPv2 pan-cancer AAC -0.15 5e-05
mRNA LAMP5 CTRPv2 pan-cancer AAC 0.14 5e-05
mRNA EWSR1 GDSC1000 pan-cancer AAC 0.12 5e-05
mRNA C1orf54 GDSC1000 pan-cancer AAC 0.13 5e-05
mRNA CLEC10A CTRPv2 pan-cancer AAC 0.13 5e-05
mRNA SNX20 CTRPv2 pan-cancer AAC 0.17 5e-05
mRNA SEC63 GDSC1000 pan-cancer AAC 0.11 6e-05
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