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YK 4-279

Synonyms

SourcesNames Used
GDSC1000, CTRPv2YK 4-279
PharmacoGx YK 4-279

External IDs

DatabaseIdentifier
Smiles: COc1ccc(cc1)C(=O)CC1(O)C(=O)Nc2c1c(Cl)ccc2Cl

Annotated Targets

EWSR1, FLI1, DHX9, ERG, ETV1

FDA Approval Status

Not Approved
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Top molecular features associated with response to YK 4-279


Feature TypeStandardized
Nominal ANOVA
mRNA MITD1 GDSC1000 pan-cancer AAC 0.2 1e-07
mRNA CEP295NL CTRPv2 pan-cancer AAC -0.2 1e-07
mRNA MAP3K4 CTRPv2 pan-cancer AAC 0.18 1e-07
mRNA WDR75 GDSC1000 pan-cancer AAC 0.19 1e-07
mRNA E2F3 CTRPv2 pan-cancer AAC 0.17 1e-07
mRNA KLHL8 CTRPv2 pan-cancer AAC 0.19 1e-07
mRNA BICDL1 GDSC1000 pan-cancer AAC -0.19 1e-07
mRNA GMEB1 CTRPv2 pan-cancer AAC 0.19 2e-07
mRNA SH2D4A CTRPv2 pan-cancer AAC -0.19 2e-07
mRNA SLC4A7 GDSC1000 pan-cancer AAC 0.19 2e-07
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