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YK 4-279

Synonyms

SourcesNames Used
GDSC1000, CTRPv2YK 4-279
PharmacoGx YK 4-279

External IDs

DatabaseIdentifier
Smiles: COc1ccc(cc1)C(=O)CC1(O)C(=O)Nc2c1c(Cl)ccc2Cl

Annotated Targets

EWSR1, FLI1, DHX9, ERG, ETV1

FDA Approval Status

Not Approved
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Top molecular features associated with response to YK 4-279


Feature TypeStandardized
Nominal ANOVA
mRNA GNG12 CTRPv2 pan-cancer AAC -0.2 1e-06
mRNA DOT1L CTRPv2 pan-cancer AAC 0.19 1e-06
mRNA SH3BP1 CTRPv2 pan-cancer AAC 0.18 1e-06
mRNA AP003419.11 CTRPv2 pan-cancer AAC -0.16 1e-06
mRNA WRN CTRPv2 pan-cancer AAC 0.16 1e-06
mRNA CAND2 CTRPv2 pan-cancer AAC 0.16 2e-06
mRNA TTC39A GDSC1000 pan-cancer AAC -0.19 2e-06
mRNA ZNF445 CTRPv2 pan-cancer AAC 0.17 2e-06
mRNA POGK CTRPv2 pan-cancer AAC 0.16 2e-06
mRNA RNF8 CTRPv2 pan-cancer AAC 0.15 2e-06
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