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GSK1070916

Synonyms

SourcesNames Used
GDSC1000, GRAYGSK1070916
PharmacoGx GSK1070916

External IDs

DatabaseIdentifier
Smiles: CCN1C=C(C(=N1)C2=CC=C(C=C2)NC(=O)N(C)C)C3=C4C=C(NC4=NC=C3)C5=CC(=CC=C5)CN(C)C
Inchikey: QTBWCSQGBMPECM-UHFFFAOYSA-N
Pubchem: 46885626

Annotated Targets

AURKA, AURKB, AURKC, CYP2D6, CYP3A4

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1070916


Feature TypeStandardized
Nominal ANOVA
mRNA HEATR5A GDSC1000 pan-cancer AAC -0.27 5e-16
mRNA CD63 GDSC1000 pan-cancer AAC -0.27 2e-12
mRNA P4HA2 GDSC1000 pan-cancer AAC -0.27 1e-11
mRNA FUCA2 GDSC1000 pan-cancer AAC -0.28 6e-15
mRNA MGAT4B GDSC1000 pan-cancer AAC -0.28 4e-14
mRNA TJP1 GDSC1000 pan-cancer AAC -0.29 1e-06
mRNA CTSA GDSC1000 pan-cancer AAC -0.29 1e-16
mRNA ITGB5 GDSC1000 pan-cancer AAC -0.29 9e-14
mRNA LGALS3 GDSC1000 pan-cancer AAC -0.3 2e-16
mRNA ATOX1 GDSC1000 pan-cancer AAC -0.3 4e-19
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