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TKI258

Synonyms

SourcesNames Used
CCLETKI258
PharmacoGx TKI258

External IDs

DatabaseIdentifier
Smiles: CN1CCN(CC1)C2=CC3=C(C=C2)NC(=C4C(=C5C(=NC4=O)C=CC=C5F)N)N3
Inchikey: KCOYQXZDFIIGCY-ZZEZOPTASA-N
Pubchem: 9886808

FDA Approval Status

Not Approved
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Top molecular features associated with response to TKI258


Feature TypeStandardized
Nominal ANOVA
mRNA RNASE3 CCLE pan-cancer AAC 0.25 8e-08
mRNA MLC1 CCLE pan-cancer AAC 0.26 1e-07
mRNA PPP1R27 CCLE pan-cancer AAC 0.24 1e-07
mRNA ASPDH CCLE pan-cancer AAC -0.24 2e-07
mRNA CCL23 CCLE pan-cancer AAC 0.24 2e-07
mRNA SERPINB10 CCLE pan-cancer AAC 0.24 3e-07
mRNA FECH CCLE pan-cancer AAC 0.24 3e-07
mRNA TIFAB CCLE pan-cancer AAC 0.23 3e-07
mRNA RAB37 CCLE pan-cancer AAC 0.27 4e-07
mRNA SRP72 CCLE pan-cancer AAC 0.24 4e-07
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