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TKI258

Synonyms

SourcesNames Used
CCLETKI258
PharmacoGx TKI258

External IDs

DatabaseIdentifier
Smiles: CN1CCN(CC1)C2=CC3=C(C=C2)NC(=C4C(=C5C(=NC4=O)C=CC=C5F)N)N3
Inchikey: KCOYQXZDFIIGCY-ZZEZOPTASA-N
Pubchem: 9886808

FDA Approval Status

Not Approved
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Top molecular features associated with response to TKI258


Feature TypeStandardized
Nominal ANOVA
mRNA PRKCB CCLE pan-cancer AAC 0.29 5e-06
mRNA SLC22A16 CCLE pan-cancer AAC 0.29 2e-09
mRNA GAPT CCLE pan-cancer AAC 0.29 2e-08
mRNA MYB CCLE pan-cancer AAC 0.3 2e-05
mRNA C1orf228 CCLE pan-cancer AAC 0.31 7e-10
mRNA DPEP2 CCLE pan-cancer AAC 0.32 2e-10
mRNA LCP2 CCLE pan-cancer AAC 0.32 3e-08
mRNA TYROBP CCLE pan-cancer AAC 0.32 1e-11
mRNA LST1 CCLE pan-cancer AAC 0.32 2e-09
mRNA GMFG CCLE pan-cancer AAC 0.33 6e-05
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