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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA LOXL2 GDSC1000 pan-cancer AAC 0.4 7e-10
mRNA C5orf46 GDSC1000 pan-cancer AAC 0.38 6e-14
mRNA CALD1 GDSC1000 pan-cancer AAC 0.37 6e-07
mRNA SPARC GDSC1000 pan-cancer AAC 0.36 2e-07
mRNA HTRA1 GDSC1000 pan-cancer AAC 0.35 3e-07
mRNA HEG1 GDSC1000 pan-cancer AAC 0.32 4e-08
mRNA FSTL1 GDSC1000 pan-cancer AAC 0.32 2e-06
mRNA THBS1 GDSC1000 pan-cancer AAC 0.32 7e-06
mRNA FAM114A1 GDSC1000 pan-cancer AAC 0.32 2e-06
mRNA WWTR1 GDSC1000 pan-cancer AAC 0.32 5e-06
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