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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA A2M GDSC1000 pan-cancer AAC 0.15 0.006
mRNA AAK1 GDSC1000 pan-cancer AAC -0.13 0.006
mRNA AAMP CTRPv2 pan-cancer AAC -0.11 0.003
mRNA ABCA3 GDSC1000 pan-cancer AAC -0.2 0.0002
mRNA ABCA6 GDSC1000 pan-cancer AAC 0.18 0.001
mRNA ABCB6 CTRPv2 pan-cancer AAC -0.11 0.006
mRNA ABCC2 GDSC1000 pan-cancer AAC 0.14 0.008
mRNA ABCC3 GDSC1000 pan-cancer AAC 0.21 0.0002
mRNA ABHD15 CTRPv2 pan-cancer AAC 0.1 0.005
mRNA ABI1 CTRPv2 pan-cancer AAC 0.12 0.002
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