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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA ZC3H12D CTRPv2 pan-cancer AAC 0.26 4e-10
mRNA FCRL1 CTRPv2 pan-cancer AAC 0.2 4e-08
mRNA PLEKHA2 CTRPv2 pan-cancer AAC 0.22 5e-08
mRNA FCRL2 CTRPv2 pan-cancer AAC 0.2 9e-08
mRNA CD79B CTRPv2 pan-cancer AAC 0.21 1e-07
mRNA MKL1 CTRPv2 pan-cancer AAC 0.2 2e-07
mRNA KANK2 CTRPv2 pan-cancer AAC 0.22 3e-07
mRNA TRAF1 CTRPv2 pan-cancer AAC 0.19 4e-07
mRNA ALOX5 CTRPv2 pan-cancer AAC 0.19 4e-07
mRNA BDH2 CTRPv2 pan-cancer AAC 0.19 7e-07
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