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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA H2AFY2 GDSC1000 pan-cancer AAC -0.26 0.0001
mRNA JAG2 GDSC1000 pan-cancer AAC -0.25 1e-05
mRNA ELAVL4 GDSC1000 pan-cancer AAC -0.22 0.001
mRNA XPO7 GDSC1000 pan-cancer AAC -0.22 6e-06
mRNA INA GDSC1000 pan-cancer AAC -0.22 0.0006
mRNA SBK1 GDSC1000 pan-cancer AAC -0.22 0.001
mRNA ICA1 GDSC1000 pan-cancer AAC -0.21 0.0009
mRNA ELAVL3 GDSC1000 pan-cancer AAC -0.21 0.001
mRNA TAGLN3 GDSC1000 pan-cancer AAC -0.21 0.0005
mRNA CHGA GDSC1000 pan-cancer AAC -0.21 0.002
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