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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA ABI3BP GDSC1000 pan-cancer AAC 0.15 0.01
mRNA ABLIM3 GDSC1000 pan-cancer AAC 0.15 0.006
mRNA ABLIM3 CTRPv2 pan-cancer AAC 0.11 0.009
mRNA AC008641.1 CTRPv2 pan-cancer AAC 0.1 0.006
mRNA AC009950.1 CTRPv2 pan-cancer AAC 0.16 3e-05
mRNA AC010412.1 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA AC011043.2 CTRPv2 pan-cancer AAC -0.094 0.01
mRNA AC013264.1 CTRPv2 pan-cancer AAC 0.14 0.002
mRNA AC019206.1 CTRPv2 pan-cancer AAC 0.12 0.001
mRNA AC022405.1 CTRPv2 pan-cancer AAC 0.14 0.0002
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