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TGX221

Synonyms

SourcesNames Used
GDSC1000TGX221
CTRPv2TGX-221
PharmacoGx TGX221

External IDs

DatabaseIdentifier
Smiles: CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Inchikey: CPRAGQJXBLMUEL-UHFFFAOYSA-N
Pubchem: 9907093

Annotated Targets

PIK3CB, PIK3CD

FDA Approval Status

Not Approved
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Top molecular features associated with response to TGX221


Feature TypeStandardized
Nominal ANOVA
mRNA ZNF706 CTRPv2 pan-cancer AAC -0.1 0.009
mRNA ZNF768 CTRPv2 pan-cancer AAC -0.11 0.004
mRNA ZNF774 CTRPv2 pan-cancer AAC -0.13 0.001
mRNA ZNF789 CTRPv2 pan-cancer AAC 0.1 0.006
mRNA ZNF804A CTRPv2 pan-cancer AAC 0.12 0.003
mRNA ZNF823 CTRPv2 pan-cancer AAC -0.1 0.01
mRNA ZNF827 GDSC1000 pan-cancer AAC 0.13 0.005
mRNA ZNF827 CTRPv2 pan-cancer AAC 0.11 0.007
mRNA ZNF830 GDSC1000 pan-cancer AAC -0.15 0.002
mRNA ZNF830 CTRPv2 pan-cancer AAC -0.11 0.006
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