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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA AMOTL2 GDSC1000 pan-cancer AAC 0.18 8e-06
mRNA SMARCC1 GDSC1000 pan-cancer AAC -0.17 8e-06
mRNA PPP1R15A GDSC1000 pan-cancer AAC 0.15 9e-06
mRNA PRR14L GDSC1000 pan-cancer AAC -0.16 1e-05
mRNA RSBN1L GDSC1000 pan-cancer AAC -0.16 1e-05
mRNA CHPF GDSC1000 pan-cancer AAC 0.16 1e-05
mRNA EXO1 GDSC1000 pan-cancer AAC -0.15 1e-05
mRNA LIG1 GDSC1000 pan-cancer AAC -0.16 1e-05
mRNA BLM GDSC1000 pan-cancer AAC -0.17 1e-05
mRNA PLEKHF1 GDSC1000 pan-cancer AAC 0.15 2e-05
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