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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA MYB GDSC1000 pan-cancer AAC -0.18 0.0002
mRNA ATAD5 GDSC1000 pan-cancer AAC -0.18 1e-06
mRNA CDC25A GDSC1000 pan-cancer AAC -0.18 3e-06
mRNA HOOK1 GDSC1000 pan-cancer AAC -0.17 2e-05
mRNA HADH GDSC1000 pan-cancer AAC -0.17 4e-06
mRNA BLM GDSC1000 pan-cancer AAC -0.17 1e-05
mRNA SMARCC1 GDSC1000 pan-cancer AAC -0.17 8e-06
mRNA PBRM1 GDSC1000 pan-cancer AAC -0.17 2e-05
mRNA RSBN1L GDSC1000 pan-cancer AAC -0.16 1e-05
mRNA MCM7 GDSC1000 pan-cancer AAC -0.16 3e-06
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