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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA TCEA3 GDSC1000 pan-cancer AAC -0.14 9e-05
mRNA POLA1 GDSC1000 pan-cancer AAC -0.14 9e-05
mRNA LITAF GDSC1000 pan-cancer AAC 0.14 9e-05
mRNA PLCXD1 GDSC1000 pan-cancer AAC -0.14 9e-05
mRNA RNH1 GDSC1000 pan-cancer AAC 0.14 0.0001
mRNA ULBP2 GDSC1000 pan-cancer AAC 0.15 0.0001
mRNA STMN1 GDSC1000 pan-cancer AAC -0.14 0.0001
mRNA CSNK1A1 GDSC1000 pan-cancer AAC 0.13 0.0001
mRNA SHC1 GDSC1000 pan-cancer AAC 0.15 0.0001
mRNA HNRNPA1L2 GDSC1000 pan-cancer AAC -0.14 0.0001
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