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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA LEO1 GDSC1000 pan-cancer AAC -0.082 0.02
mRNA AVL9 GDSC1000 pan-cancer AAC 0.083 0.02
mRNA WNT2 GDSC1000 pan-cancer AAC -0.079 0.02
mRNA CLSPN GDSC1000 pan-cancer AAC -0.083 0.02
mRNA PPP2R3B GDSC1000 pan-cancer AAC -0.083 0.02
mRNA ARPC1B GDSC1000 pan-cancer AAC 0.087 0.02
mRNA HSD11B2 GDSC1000 pan-cancer AAC -0.091 0.02
mRNA SH3GLB1 GDSC1000 pan-cancer AAC 0.083 0.02
mRNA HSPG2 GDSC1000 pan-cancer AAC 0.091 0.02
mRNA CAMKV GDSC1000 pan-cancer AAC -0.089 0.02
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