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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA LAMB2 GDSC1000 pan-cancer AAC 0.13 0.002
mRNA ASRGL1 GDSC1000 pan-cancer AAC -0.11 0.002
mRNA C9orf69 GDSC1000 pan-cancer AAC 0.11 0.002
mRNA TAF10 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA HIST1H2BF GDSC1000 pan-cancer AAC -0.11 0.002
mRNA CCNE2 GDSC1000 pan-cancer AAC -0.11 0.002
mRNA KCNJ11 GDSC1000 pan-cancer AAC -0.11 0.002
mRNA GADD45G GDSC1000 pan-cancer AAC -0.11 0.002
mRNA COX7B2 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA HACD3 GDSC1000 pan-cancer AAC -0.11 0.002
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