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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA FIBIN GDSC1000 pan-cancer AAC 0.086 0.02
mRNA PRPF40B GDSC1000 pan-cancer AAC -0.083 0.02
mRNA GIPC2 GDSC1000 pan-cancer AAC -0.088 0.02
mRNA APC2 GDSC1000 pan-cancer AAC -0.095 0.02
mRNA TTC23 GDSC1000 pan-cancer AAC 0.09 0.02
mRNA CENPK GDSC1000 pan-cancer AAC -0.082 0.02
mRNA AMOT GDSC1000 pan-cancer AAC -0.081 0.02
mRNA NRCAM GDSC1000 pan-cancer AAC -0.081 0.02
mRNA DAPK2 GDSC1000 pan-cancer AAC -0.081 0.02
mRNA KIF14 GDSC1000 pan-cancer AAC -0.08 0.02
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