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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA SLC12A4 GDSC1000 pan-cancer AAC 0.087 0.02
mRNA PGBD2 GDSC1000 pan-cancer AAC -0.085 0.02
mRNA COLCA2 GDSC1000 pan-cancer AAC -0.085 0.02
mRNA RGS3 GDSC1000 pan-cancer AAC 0.093 0.02
mRNA PAPD4 GDSC1000 pan-cancer AAC 0.098 0.02
mRNA VAC14 GDSC1000 pan-cancer AAC 0.081 0.02
mRNA TMEM39A GDSC1000 pan-cancer AAC 0.08 0.02
mRNA TFDP1 GDSC1000 pan-cancer AAC -0.085 0.02
mRNA ZFP36 GDSC1000 pan-cancer AAC 0.093 0.02
mRNA POU4F1 GDSC1000 pan-cancer AAC -0.084 0.02
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