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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA ABCC3 GDSC1000 pan-cancer AAC 0.098 0.01
mRNA LSM3 GDSC1000 pan-cancer AAC -0.087 0.01
mRNA GRAMD3 GDSC1000 pan-cancer AAC 0.097 0.01
mRNA AURKB GDSC1000 pan-cancer AAC -0.083 0.01
mRNA TRIM36 GDSC1000 pan-cancer AAC -0.083 0.01
mRNA EMC7 GDSC1000 pan-cancer AAC 0.083 0.01
mRNA STARD7 GDSC1000 pan-cancer AAC -0.09 0.01
mRNA HEXIM1 GDSC1000 pan-cancer AAC 0.086 0.01
mRNA TIGD3 GDSC1000 pan-cancer AAC -0.087 0.01
mRNA WARS GDSC1000 pan-cancer AAC 0.086 0.01
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