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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA CSRNP3 GDSC1000 pan-cancer AAC -0.095 0.01
mRNA FNDC5 GDSC1000 pan-cancer AAC -0.092 0.01
mRNA GSK3B GDSC1000 pan-cancer AAC 0.088 0.01
mRNA SMURF2 GDSC1000 pan-cancer AAC 0.093 0.01
mRNA RBMS2 GDSC1000 pan-cancer AAC 0.1 0.01
mRNA FAM83D GDSC1000 pan-cancer AAC -0.09 0.01
mRNA INTU GDSC1000 pan-cancer AAC 0.091 0.01
mRNA MYCL GDSC1000 pan-cancer AAC -0.086 0.01
mRNA ATXN7L1 GDSC1000 pan-cancer AAC -0.09 0.01
mRNA ERC2 GDSC1000 pan-cancer AAC -0.088 0.01
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