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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA UBE2QL1 GDSC1000 pan-cancer AAC -0.09 0.01
mRNA IQCC GDSC1000 pan-cancer AAC -0.087 0.01
mRNA KLHDC3 GDSC1000 pan-cancer AAC -0.091 0.01
mRNA GINS4 GDSC1000 pan-cancer AAC -0.088 0.01
mRNA ANXA5 GDSC1000 pan-cancer AAC 0.098 0.01
mRNA C17orf75 GDSC1000 pan-cancer AAC -0.085 0.01
mRNA WDR89 GDSC1000 pan-cancer AAC -0.094 0.01
mRNA PTGR1 GDSC1000 pan-cancer AAC 0.11 0.01
mRNA RUNX2 GDSC1000 pan-cancer AAC 0.09 0.01
mRNA KRIT1 GDSC1000 pan-cancer AAC -0.087 0.01
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