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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA GNAZ GDSC1000 pan-cancer AAC -0.09 0.01
mRNA SHISA4 GDSC1000 pan-cancer AAC 0.11 0.01
mRNA ARNTL2 GDSC1000 pan-cancer AAC 0.097 0.01
mRNA PLPP1 GDSC1000 pan-cancer AAC 0.093 0.01
mRNA NFAT5 GDSC1000 pan-cancer AAC 0.09 0.01
mRNA WNT7B GDSC1000 pan-cancer AAC 0.098 0.01
mRNA IP6K2 GDSC1000 pan-cancer AAC -0.09 0.01
mRNA SLC35F1 GDSC1000 pan-cancer AAC -0.096 0.01
mRNA CASP8AP2 GDSC1000 pan-cancer AAC -0.091 0.01
mRNA GPC2 GDSC1000 pan-cancer AAC -0.098 0.01
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