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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA ZNF530 GDSC1000 pan-cancer AAC -0.087 0.009
mRNA NDC80 GDSC1000 pan-cancer AAC -0.091 0.009
mRNA ABLIM2 GDSC1000 pan-cancer AAC -0.089 0.009
mRNA FAM76B GDSC1000 pan-cancer AAC -0.099 0.009
mRNA ENTPD8 GDSC1000 pan-cancer AAC -0.089 0.009
mRNA LMNB1 GDSC1000 pan-cancer AAC -0.095 0.009
mRNA NKX2-2 GDSC1000 pan-cancer AAC -0.11 0.009
mRNA MEIS1 GDSC1000 pan-cancer AAC -0.099 0.009
mRNA RRM1 GDSC1000 pan-cancer AAC -0.088 0.009
mRNA RNF144A GDSC1000 pan-cancer AAC -0.099 0.009
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