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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA KRT81 GDSC1000 pan-cancer AAC 0.12 0.0008
mRNA E2F2 GDSC1000 pan-cancer AAC -0.13 0.0008
mRNA ALG2 GDSC1000 pan-cancer AAC 0.11 0.0008
mRNA IFNA2 GDSC1000 pan-cancer AAC 0.11 0.0008
mRNA TOP2A GDSC1000 pan-cancer AAC -0.11 0.0008
mRNA POLE2 GDSC1000 pan-cancer AAC -0.12 0.0008
mRNA CENPF GDSC1000 pan-cancer AAC -0.11 0.0008
mRNA CA12 GDSC1000 pan-cancer AAC 0.12 0.0008
mRNA GUSB GDSC1000 pan-cancer AAC -0.12 0.0009
mRNA CDCA7 GDSC1000 pan-cancer AAC -0.12 0.0009
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