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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA INPP5J GDSC1000 pan-cancer AAC -0.12 0.0008
mRNA COL21A1 GDSC1000 pan-cancer AAC -0.12 0.0008
mRNA C2CD5 GDSC1000 pan-cancer AAC -0.12 0.0008
mRNA ZWILCH GDSC1000 pan-cancer AAC -0.11 0.0008
mRNA OSTF1 GDSC1000 pan-cancer AAC 0.14 0.0008
mRNA RFC4 GDSC1000 pan-cancer AAC -0.12 0.0008
mRNA CBX1 GDSC1000 pan-cancer AAC -0.12 0.0008
mRNA UBTF GDSC1000 pan-cancer AAC -0.12 0.0008
mRNA GNG12 GDSC1000 pan-cancer AAC 0.17 0.0008
mRNA BCL9L GDSC1000 pan-cancer AAC 0.14 0.0008
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