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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA TMEM240 GDSC1000 pan-cancer AAC -0.082 0.02
mRNA ANKS4B GDSC1000 pan-cancer AAC -0.094 0.02
mRNA CNTN3 GDSC1000 pan-cancer AAC -0.081 0.02
mRNA LRRC43 GDSC1000 pan-cancer AAC -0.08 0.02
mRNA P3H4 GDSC1000 pan-cancer AAC 0.1 0.02
mRNA KMT2D GDSC1000 pan-cancer AAC -0.087 0.02
mRNA HMGCS1 GDSC1000 pan-cancer AAC -0.082 0.02
mRNA ATP23 GDSC1000 pan-cancer AAC -0.097 0.02
mRNA CELF5 GDSC1000 pan-cancer AAC -0.087 0.02
mRNA PHF8 GDSC1000 pan-cancer AAC -0.089 0.02
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