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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA FAM214B GDSC1000 pan-cancer AAC 0.15 4e-05
mRNA CREB3 GDSC1000 pan-cancer AAC 0.14 4e-05
mRNA TRIOBP GDSC1000 pan-cancer AAC 0.15 4e-05
mRNA PBK GDSC1000 pan-cancer AAC -0.14 4e-05
mRNA KNTC1 GDSC1000 pan-cancer AAC -0.15 4e-05
mRNA SDC4 GDSC1000 pan-cancer AAC 0.2 5e-05
mRNA TNKS1BP1 GDSC1000 pan-cancer AAC 0.16 5e-05
mRNA KIF11 GDSC1000 pan-cancer AAC -0.14 5e-05
mRNA PXN GDSC1000 pan-cancer AAC 0.16 5e-05
mRNA EPB41 GDSC1000 pan-cancer AAC -0.16 5e-05
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