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FTI-277

Synonyms

SourcesNames Used
GDSC1000FTI-277
PharmacoGx FTI-277

External IDs

DatabaseIdentifier
Smiles: COC(=O)C(CCSC)NC(=O)C1=C(C=C(C=C1)NCC(CS)N)C2=CC=CC=C2
Inchikey: GKFPROVOIQKYTO-UZLBHIALSA-N
Pubchem: 3005532

FDA Approval Status

Not Approved
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Top molecular features associated with response to FTI-277


Feature TypeStandardized
Nominal ANOVA
mRNA FANCD2 GDSC1000 pan-cancer AAC -0.15 7e-05
mRNA UBE2H GDSC1000 pan-cancer AAC 0.14 7e-05
mRNA TIMM13 GDSC1000 pan-cancer AAC -0.14 7e-05
mRNA LGALS1 GDSC1000 pan-cancer AAC 0.15 7e-05
mRNA PPIC GDSC1000 pan-cancer AAC 0.19 7e-05
mRNA PDIK1L GDSC1000 pan-cancer AAC -0.15 7e-05
mRNA EFR3A GDSC1000 pan-cancer AAC 0.14 7e-05
mRNA TNFRSF10B GDSC1000 pan-cancer AAC 0.14 8e-05
mRNA HSPA14 GDSC1000 pan-cancer AAC -0.14 8e-05
mRNA DRAP1 GDSC1000 pan-cancer AAC 0.14 8e-05
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